{"id":950,"date":"2023-05-27T14:40:15","date_gmt":"2023-05-27T14:40:15","guid":{"rendered":"https:\/\/dailyai.com\/?p=950"},"modified":"2023-06-01T09:26:45","modified_gmt":"2023-06-01T09:26:45","slug":"ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria","status":"publish","type":"post","link":"https:\/\/dailyai.com\/sv\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/","title":{"rendered":"AI uppt\u00e4cker ny antibiotika f\u00f6r l\u00e4kemedelsresistenta bakterier"},"content":{"rendered":"<p><b>M\u00e4nskligheten har hamnat p\u00e5 efterk\u00e4lken i kampen mot l\u00e4kemedelsresistenta bakterier, men AI kan visa sig vara v\u00e5rt hemliga vapen.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400\">Antibiotikaresistenta patogener \u00e4r ansvariga f\u00f6r mellan <\/span><a href=\"https:\/\/www.thelancet.com\/journals\/lancet\/article\/PIIS0140-6736(21)02724-0\/fulltext\"><span style=\"font-weight: 400\">1 och 5 miljoner d\u00f6dsfall<\/span><\/a><span style=\"font-weight: 400\"> per \u00e5r.\u00a0\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">F\u00e5 nya antibiotika har tagits fram under det senaste decenniet, och de flesta \u00e4r sm\u00e5 justeringar av befintliga antibiotika.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Att uppt\u00e4cka nya l\u00e4kemedel \u00e4r exceptionellt arbetsintensivt, men en ny banbrytande studie har utnyttjat AI f\u00f6r att automatiskt screena tusentals f\u00f6reningar f\u00f6r att uppt\u00e4cka v\u00e4gar f\u00f6r laboratorietester.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Den <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41589-023-01349-8.epdf?sharing_token=8HV9JdX6i-6DpHj0fv2wOtRgN0jAjWel9jnR3ZoTv0PgqDK_eQp8NcAST1F90jpq3WEGXG2Su3RGayoL_4HVm-885WktBHURHlCxulwlcvqKkHgdWqrHo6v6OktzRXc-zL4MsysGdAFnKBAI2wyymCj5gtw5qVJSvyZDrTK_wGIpI8eaOx1jqmIvwv1jdlYBYoAQi8TfYbpGh2Cfrhw5BG1rJNzyE_FFkgm1zzQdwpc%3D&amp;tracking_referrer=www.bbc.co.uk\"><span style=\"font-weight: 400\">studie<\/span><\/a><span style=\"font-weight: 400\">som publicerades i Nature Chemical Biology, f\u00f6rs\u00f6kte forskare fr\u00e5n MIT och McMaster University uppt\u00e4cka nya l\u00e4kemedel f\u00f6r att d\u00f6da<\/span><i><span style=\"font-weight: 400\"> Acinetobacter baumannii<\/span><\/i><span style=\"font-weight: 400\">, en bakterie som <\/span><a href=\"https:\/\/www.who.int\/news\/item\/27-02-2017-who-publishes-list-of-bacteria-for-which-new-antibiotics-are-urgently-needed\"><span style=\"font-weight: 400\">WHO identifierade<\/span><\/a><span style=\"font-weight: 400\"> som ett \"kritiskt hot\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">Forskarna anv\u00e4nde tv\u00e5 modeller f\u00f6r maskininl\u00e4rning (ML) f\u00f6r att automatisera processen f\u00f6r l\u00e4kemedelsuppt\u00e4ckt <\/span><a href=\"https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC1978274\/\"><i><span style=\"font-weight: 400\">in silico<\/span><\/i><\/a><span style=\"font-weight: 400\">vilket betyder \"i en dator\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">S\u00e5 h\u00e4r gick det till:<\/span><\/p>\n<p><b>Erh\u00e5llna tr\u00e4ningsdata<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Forskarna exponerade laboratorieodlade <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\"> till cirka 7 500 olika kemiska f\u00f6reningar och \u00f6vervakades f\u00f6r att se vilka f\u00f6reningar som h\u00e4mmade mikrobens tillv\u00e4xt.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">De kemiska strukturerna f\u00f6r dem som h\u00e4mmade tillv\u00e4xten matades in i en maskininl\u00e4rningsmodell (ML). Detta gjorde det m\u00f6jligt f\u00f6r modellen att l\u00e4ra sig de kemiska egenskaper som \u00e4r f\u00f6rknippade med tillv\u00e4xth\u00e4mning.<\/span><\/li>\n<\/ul>\n<p><b>Utbildat och testat modellen<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">N\u00e4r modellen hade tr\u00e4nats anv\u00e4nde forskarna den f\u00f6r att analysera en upps\u00e4ttning av 6.680 f\u00f6reningar som modellen inte tidigare hade st\u00f6tt p\u00e5. Dessa f\u00f6reningar h\u00e4mtades fr\u00e5n Drug Repurposing Hub vid Broad Institute. Den valde ut n\u00e5gra hundra f\u00f6reningar.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Forskarna valde ut 240 av dessa f\u00f6r att testa dem experimentellt i laboratoriet.\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">De fokuserade p\u00e5 f\u00f6reningar med olika strukturer j\u00e4mf\u00f6rt med befintliga antibiotika, eftersom detta g\u00f6r dem mer ben\u00e4gna att undvika antibiotikaresistens.\u00a0<\/span><\/li>\n<\/ul>\n<p><b>Experimentell laboratorietestning<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Labbtester begr\u00e4nsade listan till 9 antibiotika.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Bland dessa visade sig en f\u00f6rening som ursprungligen unders\u00f6ktes som ett potentiellt diabetesl\u00e4kemedel vara extremt effektiv f\u00f6r att d\u00f6da <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\">. L\u00e4kemedlet kallades \"abaucin\".\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">M\u00e4rkligt nog p\u00e5verkade det inte andra bakteriearter, inklusive <\/span><i><span style=\"font-weight: 400\">Pseudomonas aeruginosa, Staphylococcus aureus, <\/span><\/i><span style=\"font-weight: 400\">och <\/span><i><span style=\"font-weight: 400\">Enterobacteriaceae.<\/span><\/i><\/li>\n<\/ul>\n<p><span style=\"font-weight: 400\">Dr. Stokes, som arbetade med projektet, <\/span><a href=\"https:\/\/www.bbc.co.uk\/news\/health-65709834\"><span style=\"font-weight: 400\">ber\u00e4ttade f\u00f6r BBC<\/span><\/a><span style=\"font-weight: 400\">\"Det \u00e4r nu arbetet b\u00f6rjar.\"\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Antibiotikan kommer att genomg\u00e5 en l\u00e5ngvarig testprocedur f\u00f6r att bed\u00f6ma dess s\u00e4kerhet i m\u00e4nniskor, vilket kanske inte \u00e4r klart f\u00f6rr\u00e4n 2030.<\/span><\/p>\n<p><span style=\"font-weight: 400\">Trots detta p\u00e5skyndar AI den arbetsintensiva uppgiften att utforska nya l\u00e4kemedel och hj\u00e4lper forskare att uppt\u00e4cka intressanta och nya antimikrobiella f\u00f6reningar. M\u00e5nga av dem har utvecklats f\u00f6r andra \u00e4ndam\u00e5l, s\u00e5 de finns redan d\u00e4r ute - vi beh\u00f6ver bara hitta dem.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Dr. Stokes sa: \"AI \u00f6kar takten, och i en perfekt v\u00e4rld minskar kostnaden, med vilken vi kan uppt\u00e4cka dessa nya klasser av antibiotika som vi desperat beh\u00f6ver.\"\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">\u00c4ven om det fortfarande \u00e4r en l\u00e5ngsam process att testa s\u00e4kerheten hos m\u00e4nniskor kommer AI-st\u00f6dda forskningspipelines s\u00e4kerligen att p\u00e5skynda marknadsintroduktionen f\u00f6r antibiotika och andra l\u00e4kemedel. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>M\u00e4nskligheten har hamnat p\u00e5 efterk\u00e4lken i kampen mot l\u00e4kemedelsresistenta bakterier, men AI kan visa sig vara v\u00e5rt hemliga vapen.  Antibiotikaresistenta patogener \u00e4r ansvariga f\u00f6r mellan 1 och 5 miljoner d\u00f6dsfall per \u00e5r.   F\u00e5 nya antibiotika har utvecklats under det senaste decenniet, och de flesta \u00e4r sm\u00e5 justeringar av befintliga antibiotika.  Att uppt\u00e4cka nya l\u00e4kemedel \u00e4r exceptionellt arbetsintensivt, men en ny banbrytande studie har utnyttjat AI f\u00f6r att automatiskt screena tusentals f\u00f6reningar f\u00f6r att uppt\u00e4cka v\u00e4gar f\u00f6r laboratorietestning.  I studien, som publicerades i Nature Chemical Biology, f\u00f6rs\u00f6kte forskare fr\u00e5n MIT och McMaster University uppt\u00e4cka nya l\u00e4kemedel f\u00f6r att d\u00f6da Acinetobacter baumannii,<\/p>","protected":false},"author":2,"featured_media":951,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[105,101],"class_list":["post-950","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI discovers new antibiotic for drug-resistant bacteria | DailyAI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" 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