{"id":8436,"date":"2023-12-19T16:35:20","date_gmt":"2023-12-19T16:35:20","guid":{"rendered":"https:\/\/dailyai.com\/?p=8436"},"modified":"2023-12-19T16:35:20","modified_gmt":"2023-12-19T16:35:20","slug":"ai-designed-proteins-display-exceptional-binding-strengths","status":"publish","type":"post","link":"https:\/\/dailyai.com\/sv\/2023\/12\/ai-designed-proteins-display-exceptional-binding-strengths\/","title":{"rendered":"AI-designade proteiner uppvisar exceptionella bindningsstyrkor"},"content":{"rendered":"<p><strong>Forskare vid University of Washington School of Medicine anv\u00e4nde AI f\u00f6r att designa nya proteinmolekyler p\u00e5 ett s\u00e4tt som \u00f6ppnar sp\u00e4nnande m\u00f6jligheter f\u00f6r uppt\u00e4ckt och behandling av sjukdomar.<\/strong><\/p>\n<p>Hur effektivt ett l\u00e4kemedel \u00e4r vid behandling av en sjukdom beror till stor del p\u00e5 hur specifikt det binder till det sjukdomsframkallande m\u00e5let och hur starkt det binder till m\u00e5let.<\/p>\n<p>Den n\u00e4stan o\u00e4ndliga m\u00e4ngden potentiella proteinformer g\u00f6r det till en extremt sv\u00e5r uppgift att designa ett protein med b\u00e5de h\u00f6g affinitet (bindningsstyrka) och h\u00f6g specificitet.<\/p>\n<p>Att hitta proteiner som binder starkt till helikala peptidm\u00e5l som glukagon, neuropeptid Y och parathormon var den utmanande uppgift som forskarna hoppades att AI skulle kunna hj\u00e4lpa till med. Deras papper, <a href=\"https:\/\/www.nature.com\/articles\/s41586-023-06953-1\" target=\"_blank\" rel=\"noopener\">publicerad i Nature<\/a>visar potentialen f\u00f6r AI att revolutionera <a href=\"https:\/\/dailyai.com\/sv\/2023\/12\/astrazeneca-bets-247m-on-ai-company-developing-cancer-drug\/\">l\u00e4kemedelsutveckling<\/a>.<\/p>\n<p>Forskarna anv\u00e4nde f\u00f6rst hallucinationsmetoder f\u00f6r djupinl\u00e4rning med AlphaFold2 och RosettaFold. Dessa avancerade AI-program har varit till stor hj\u00e4lp vid utformningen av nya proteiner, men de anv\u00e4nder mycket datorkraft.<\/p>\n<p>I ett f\u00f6rs\u00f6k att hitta en mer ber\u00e4kningseffektiv metod f\u00f6r proteindesign v\u00e4nde sig forskarna till ett tillv\u00e4gag\u00e5ngss\u00e4tt som liknar det som driver AI-bildgeneratormodeller som Stable Diffusion och DALL-E.<\/p>\n<blockquote class=\"twitter-tweet\">\n<p dir=\"ltr\" lang=\"en\">Tidningen idag <a href=\"https:\/\/twitter.com\/Nature?ref_src=twsrc%5Etfw\">@Natur<\/a> beskriver <a href=\"https:\/\/twitter.com\/UWproteindesign?ref_src=twsrc%5Etfw\">@UWproteindesign<\/a> AI-genererat protein med exceptionellt h\u00f6g bindningsaffinitet och specificitet. Denna bioteknik har betydelse f\u00f6r l\u00e4kemedelsutveckling, sjukdomsdetektering och milj\u00f6\u00f6vervakning. <a href=\"https:\/\/t.co\/KhtGhiyf6I\">https:\/\/t.co\/KhtGhiyf6I<\/a><\/p>\n<p>- UW Medicine Newsroom (@uwmnewsroom) <a href=\"https:\/\/twitter.com\/uwmnewsroom\/status\/1736785659137016153?ref_src=twsrc%5Etfw\">18 december 2023<\/a><\/p><\/blockquote>\n<p><script async src=\"https:\/\/platform.twitter.com\/widgets.js\" charset=\"utf-8\"><\/script><\/p>\n<h2>RF-diffusion<\/h2>\n<p>RFdiffusion \u00e4r en banbrytande generativ AI-modell som tr\u00e4nas p\u00e5 data fr\u00e5n k\u00e4nda proteinstrukturer. Modellen f\u00f6rfinar och omorganiserar sedan iterativt atomer till definierade proteinstrukturer.<\/p>\n<p>RFdiffusion tr\u00e4nades f\u00f6r att iterativt ta bort brus fr\u00e5n moln av fr\u00e5nkopplade atomer och sedan ordna om dem till nya proteinstrukturer. Denna modell anv\u00e4ndes tillsammans med programvaruverktyget ProteinMPNN som utformats av Baker Lab, en del av <a href=\"https:\/\/www.ipd.uw.edu\/\" target=\"_blank\" rel=\"noopener\">Institutet f\u00f6r proteindesign<\/a> vid University of Washington.<\/p>\n<p>ProteinMPNN tar en proteinstruktur som indata och anv\u00e4nder deep learning-tekniker f\u00f6r att snabbt identifiera nya aminosyrasekvenser som sannolikt kommer att vikas till specifika proteinstrukturer.<\/p>\n<h2>Sp\u00e4nnande resultat<\/h2>\n<p>De proteiner som forskarna utformade uppvisade exceptionellt h\u00f6g affinitet och specificitet f\u00f6r de peptider som de var inriktade p\u00e5. Detta inneb\u00e4r att de potentiellt skulle kunna anv\u00e4ndas f\u00f6r att skapa l\u00e4kemedel som riktar sig mot orsaken till en sjukdom snarare \u00e4n att binda till oavsiktliga m\u00e5l och potentiellt orsaka biverkningar.<\/p>\n<p>Proteinsyntes \u00e4r inget nytt, men den h\u00e4r nya metoden levererade proteiner som uppn\u00e5dde den h\u00f6gsta interaktionsstyrka som n\u00e5gonsin rapporterats mellan en biomolekyl som designats av en dator och dess m\u00e5l.<\/p>\n<p>David Baker, professor i biokemi vid UW Medicine och utredare vid Howard Hughes Medical Institute, var huvudf\u00f6rfattare till forskningsrapporten.<\/p>\n<p>Baker f\u00f6rklarade betydelsen av resultaten med att s\u00e4ga: \"M\u00f6jligheten att generera nya proteiner med s\u00e5 h\u00f6g bindningsaffinitet och specificitet \u00f6ppnar upp en v\u00e4rld av m\u00f6jligheter, fr\u00e5n nya sjukdomsbehandlingar till avancerad diagnostik.\"<\/p>\n<p>Det finns m\u00e5nga sjukdomar som idag behandlas med hj\u00e4lp av antikroppar. Antikroppar \u00e4r dock dyra att producera och har inte s\u00e4rskilt l\u00e5ng h\u00e5llbarhet.<\/p>\n<p>Preetham Venkatesh, en av de ledande forskarna, s\u00e4ger: \"Det finns m\u00e5nga sjukdomar som \u00e4r sv\u00e5ra att behandla idag helt enkelt f\u00f6r att det \u00e4r s\u00e5 utmanande att uppt\u00e4cka vissa molekyler i kroppen. Som diagnosverktyg kan designade proteiner vara ett mer kostnadseffektivt alternativ till antikroppar.\"<\/p>\n<p>Forskarna kunde validera sina biodesignmetoder genom att utf\u00f6ra laboratorietester i samarbete med Joseph Rogers Lab vid K\u00f6penhamns universitet och Andrew Hoofnagle Lab vid UW Medicine.<\/p>\n<p>Forskningen \u00e4r ett bra exempel p\u00e5 hur AI p\u00e5skyndar utvecklingen av nya behandlingar f\u00f6r sjukdomar. Artikeln \u00e4r \u00e4nnu inte peer-review-granskad men de f\u00f6rsta resultaten \u00e4r mycket sp\u00e4nnande.<\/p>","protected":false},"excerpt":{"rendered":"<p>Forskare vid University of Washington School of Medicine anv\u00e4nde AI f\u00f6r att designa nya proteinmolekyler p\u00e5 ett s\u00e4tt som \u00f6ppnar upp sp\u00e4nnande m\u00f6jligheter f\u00f6r uppt\u00e4ckt och behandling av sjukdomar. Hur effektivt ett l\u00e4kemedel \u00e4r f\u00f6r att behandla en sjukdom beror till stor del p\u00e5 hur specifikt det binder till det sjukdomsframkallande m\u00e5let och hur starkt det binder till m\u00e5let. Den n\u00e4stan o\u00e4ndliga m\u00e4ngden potentiella proteinformer g\u00f6r det till en extremt sv\u00e5r uppgift att designa ett protein med b\u00e5de h\u00f6g affinitet (bindningsstyrka) och h\u00f6g specificitet. Att hitta proteiner som binder starkt till helikala peptidm\u00e5l som glukagon, neuropeptid Y och parathyroid<\/p>","protected":false},"author":6,"featured_media":8468,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[150,203,101],"class_list":["post-8436","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-ai-benefits","tag-biotech","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI-designed proteins display exceptional binding strengths | DailyAI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/dailyai.com\/sv\/2023\/12\/ai-designed-proteins-display-exceptional-binding-strengths\/\" \/>\n<meta property=\"og:locale\" content=\"sv_SE\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"AI-designed proteins display exceptional binding strengths | DailyAI\" \/>\n<meta property=\"og:description\" content=\"Scientists at the University of Washington School of Medicine used AI to design new protein molecules in a way that opens up exciting possibilities for the detection and treatment of diseases. The effectiveness of a drug in treating a disease depends largely on how specific it is in attaching to the disease-causing target, and how strongly it attaches to the target. The near-infinite amount of potential protein shapes makes designing a protein with both high affinity (binding strength) and high specificity an extremely difficult task. 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