{"id":950,"date":"2023-05-27T14:40:15","date_gmt":"2023-05-27T14:40:15","guid":{"rendered":"https:\/\/dailyai.com\/?p=950"},"modified":"2023-06-01T09:26:45","modified_gmt":"2023-06-01T09:26:45","slug":"ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria","status":"publish","type":"post","link":"https:\/\/dailyai.com\/pt\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/","title":{"rendered":"IA descobre novo antibi\u00f3tico para bact\u00e9rias resistentes a medicamentos"},"content":{"rendered":"<p><b>A humanidade ficou para tr\u00e1s na luta contra as bact\u00e9rias resistentes aos medicamentos, mas a IA pode vir a ser a nossa arma secreta.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400\">Os agentes patog\u00e9nicos resistentes aos antibi\u00f3ticos s\u00e3o respons\u00e1veis por entre <\/span><a href=\"https:\/\/www.thelancet.com\/journals\/lancet\/article\/PIIS0140-6736(21)02724-0\/fulltext\"><span style=\"font-weight: 400\">1 e 5 milh\u00f5es de mortes<\/span><\/a><span style=\"font-weight: 400\"> por ano.\u00a0\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Poucos novos antibi\u00f3ticos foram desenvolvidos na \u00faltima d\u00e9cada e a maioria s\u00e3o ligeiras altera\u00e7\u00f5es aos antibi\u00f3ticos existentes.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">A descoberta de novos f\u00e1rmacos \u00e9 excecionalmente trabalhosa, mas um estudo recente de refer\u00eancia utilizou a IA para analisar automaticamente milhares de compostos e descobrir pistas para testes em laborat\u00f3rio.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">O <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41589-023-01349-8.epdf?sharing_token=8HV9JdX6i-6DpHj0fv2wOtRgN0jAjWel9jnR3ZoTv0PgqDK_eQp8NcAST1F90jpq3WEGXG2Su3RGayoL_4HVm-885WktBHURHlCxulwlcvqKkHgdWqrHo6v6OktzRXc-zL4MsysGdAFnKBAI2wyymCj5gtw5qVJSvyZDrTK_wGIpI8eaOx1jqmIvwv1jdlYBYoAQi8TfYbpGh2Cfrhw5BG1rJNzyE_FFkgm1zzQdwpc%3D&amp;tracking_referrer=www.bbc.co.uk\"><span style=\"font-weight: 400\">estudo<\/span><\/a><span style=\"font-weight: 400\">publicada na revista Nature Chemical Biology, investigadores do MIT e da Universidade McMaster tentaram descobrir novos medicamentos para matar<\/span><i><span style=\"font-weight: 400\"> Acinetobacter baumannii<\/span><\/i><span style=\"font-weight: 400\">, uma bact\u00e9ria a <\/span><a href=\"https:\/\/www.who.int\/news\/item\/27-02-2017-who-publishes-list-of-bacteria-for-which-new-antibiotics-are-urgently-needed\"><span style=\"font-weight: 400\">A OMS identificou<\/span><\/a><span style=\"font-weight: 400\"> como uma \"amea\u00e7a cr\u00edtica\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">Os investigadores utilizaram dois modelos de aprendizagem autom\u00e1tica (ML) para automatizar o processo de descoberta de medicamentos <\/span><a href=\"https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC1978274\/\"><i><span style=\"font-weight: 400\">in silico<\/span><\/i><\/a><span style=\"font-weight: 400\">, que significa \"num computador\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">Eis como funcionava:<\/span><\/p>\n<p><b>Dados de treino obtidos<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Os investigadores expuseram <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\"> a cerca de 7.500 compostos qu\u00edmicos diferentes e monitorizados para ver quais os compostos que inibiam o crescimento do micr\u00f3bio.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">As estruturas qu\u00edmicas das subst\u00e2ncias que inibiam o crescimento foram introduzidas num modelo de aprendizagem autom\u00e1tica (ML). Isto permitiu que o modelo aprendesse as caracter\u00edsticas qu\u00edmicas associadas \u00e0 inibi\u00e7\u00e3o do crescimento.<\/span><\/li>\n<\/ul>\n<p><b>Treinou e testou o modelo<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Uma vez treinado o modelo, os investigadores utilizaram-no para analisar um conjunto de 6.680 compostos que o modelo n\u00e3o tinha encontrado anteriormente. Estes compostos foram obtidos no Drug Repurposing Hub do Broad Institute. O modelo seleccionou algumas centenas de compostos.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Os investigadores escolheram 240 da lista restrita para testar experimentalmente no laborat\u00f3rio.\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Concentraram-se em compostos com estruturas diferenciadas dos antibi\u00f3ticos existentes, uma vez que isso os torna mais suscept\u00edveis de escapar \u00e0 resist\u00eancia aos antibi\u00f3ticos.\u00a0<\/span><\/li>\n<\/ul>\n<p><b>Ensaios laboratoriais experimentais<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Os testes laboratoriais reduziram a lista a 9 antibi\u00f3ticos.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Entre estes, um composto inicialmente explorado como um potencial medicamento para a diabetes revelou-se extremamente eficaz para matar <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\">. O medicamento chamava-se \"abaucin\".\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Peculiarmente, n\u00e3o afectou outras esp\u00e9cies de bact\u00e9rias, incluindo <\/span><i><span style=\"font-weight: 400\">Pseudomonas aeruginosa, Staphylococcus aureus, <\/span><\/i><span style=\"font-weight: 400\">e <\/span><i><span style=\"font-weight: 400\">Enterobacteriaceae.<\/span><\/i><\/li>\n<\/ul>\n<p><span style=\"font-weight: 400\">Dr. Stokes, que trabalhou no projeto, <\/span><a href=\"https:\/\/www.bbc.co.uk\/news\/health-65709834\"><span style=\"font-weight: 400\">disse \u00e0 BBC<\/span><\/a><span style=\"font-weight: 400\">\"\u00c9 agora que o trabalho come\u00e7a\".\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">O antibi\u00f3tico ser\u00e1 submetido a um longo processo de testes para avaliar a sua seguran\u00e7a nos seres humanos, que poder\u00e1 n\u00e3o estar conclu\u00eddo antes de 2030.<\/span><\/p>\n<p><span style=\"font-weight: 400\">Mesmo assim, a IA acelera a tarefa trabalhosa de explorar novos medicamentos, ajudando os investigadores a descobrir compostos antimicrobianos novos e interessantes. Muitos j\u00e1 foram desenvolvidos para outros fins, por isso j\u00e1 existem - s\u00f3 precisamos de os encontrar.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Segundo o Dr. Stokes, \"a IA aumenta a taxa e, num mundo perfeito, diminui o custo com que podemos descobrir estas novas classes de antibi\u00f3ticos de que precisamos desesperadamente\".\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Embora o teste de seguran\u00e7a em humanos continue a ser um processo lento, as linhas de investiga\u00e7\u00e3o apoiadas pela IA ir\u00e3o certamente acelerar o tempo de coloca\u00e7\u00e3o no mercado de antibi\u00f3ticos e outros produtos farmac\u00eauticos. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>A humanidade ficou para tr\u00e1s na luta contra as bact\u00e9rias resistentes aos medicamentos, mas a IA pode vir a ser a nossa arma secreta.  Os agentes patog\u00e9nicos resistentes aos antibi\u00f3ticos s\u00e3o respons\u00e1veis por 1 a 5 milh\u00f5es de mortes por ano.   Na \u00faltima d\u00e9cada, foram desenvolvidos poucos antibi\u00f3ticos novos e a maioria s\u00e3o ligeiras altera\u00e7\u00f5es aos antibi\u00f3ticos existentes.  A descoberta de novos f\u00e1rmacos \u00e9 excecionalmente trabalhosa, mas um estudo recente e marcante aproveitou a IA para analisar automaticamente milhares de compostos e descobrir pistas para testes em laborat\u00f3rio.  No estudo, publicado na revista Nature Chemical Biology, investigadores do MIT e da Universidade McMaster tentaram descobrir novos f\u00e1rmacos para matar a bact\u00e9ria Acinetobacter baumannii,<\/p>","protected":false},"author":2,"featured_media":951,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[105,101],"class_list":["post-950","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI discovers new antibiotic for drug-resistant bacteria | DailyAI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" 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