{"id":2384,"date":"2023-07-07T20:16:06","date_gmt":"2023-07-07T20:16:06","guid":{"rendered":"https:\/\/dailyai.com\/?p=2384"},"modified":"2023-07-07T21:05:18","modified_gmt":"2023-07-07T21:05:18","slug":"ai-accelerates-discovery-of-anti-aging-drugs-in-new-study","status":"publish","type":"post","link":"https:\/\/dailyai.com\/pt\/2023\/07\/ai-accelerates-discovery-of-anti-aging-drugs-in-new-study\/","title":{"rendered":"IA acelera a descoberta de medicamentos anti-envelhecimento num novo estudo"},"content":{"rendered":"<p><b>Uma equipa internacional de investigadores da Universidade de Edimburgo e do Conselho Nacional de Investiga\u00e7\u00e3o espanhol IBBTEC-CSIC utilizou a IA para acelerar a descoberta de medicamentos anti-envelhecimento.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400;\">Os seus <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41467-023-39120-1\"><span style=\"font-weight: 400;\">estudo<\/span><\/a><span style=\"font-weight: 400;\"> identificaram 3 potenciais medicamentos senol\u00edticos capazes de desacelerar o envelhecimento e prevenir doen\u00e7as relacionadas com a idade. Estes medicamentos funcionam eliminando as c\u00e9lulas senescentes, frequentemente designadas por \"c\u00e9lulas zombie\". Estas c\u00e9lulas permanecem metabolicamente activas, mas s\u00e3o incapazes de se replicar.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Embora a paragem da replica\u00e7\u00e3o celular funcione como um mecanismo de defesa para evitar a propaga\u00e7\u00e3o de danos celulares, n\u00e3o \u00e9 totalmente simples.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Esta medida de prote\u00e7\u00e3o destina-se principalmente a impedir a prolifera\u00e7\u00e3o de c\u00e9lulas que sofreram danos no ADN - por exemplo, c\u00e9lulas que foram prejudicadas pela exposi\u00e7\u00e3o \u00e0 luz solar. Ao travar a replica\u00e7\u00e3o destas c\u00e9lulas danificadas, o organismo garante que estes danos n\u00e3o se propagam a outras c\u00e9lulas.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">No entanto, estas c\u00e9lulas que pararam de se dividir, conhecidas como c\u00e9lulas senescentes, podem potencialmente causar danos. Quando entram na fase de senesc\u00eancia, come\u00e7am a libertar prote\u00ednas conhecidas por causarem inflama\u00e7\u00e3o.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Isto pode afetar as c\u00e9lulas saud\u00e1veis vizinhas, criando potencialmente um ambiente inflamat\u00f3rio.\u00a0<\/span><span style=\"font-weight: 400;\">Com o tempo, esta acumula\u00e7\u00e3o de inflama\u00e7\u00e3o pode contribuir para v\u00e1rias complica\u00e7\u00f5es de sa\u00fade.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Por exemplo, a inflama\u00e7\u00e3o est\u00e1 associada a muitas doen\u00e7as, incluindo doen\u00e7as neurol\u00f3gicas e degenerativas, diabetes tipo 2, fibrose pulmonar, osteoartrite e cancro.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Por conseguinte, embora a paragem da replica\u00e7\u00e3o celular seja crucial para evitar a propaga\u00e7\u00e3o de danos no ADN, a resposta inflamat\u00f3ria associada \u00e0s c\u00e9lulas senescentes pode conduzir a outros problemas de sa\u00fade se n\u00e3o for devidamente gerida.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">E \u00e9 a\u00ed que os medicamentos senol\u00edticos podem ajudar.\u00a0<\/span><\/p>\n<h2><span style=\"font-weight: 400;\">O papel da IA<\/span><\/h2>\n<p><span style=\"font-weight: 400;\">Investiga\u00e7\u00f5es anteriores em ratos de laborat\u00f3rio demonstraram que os medicamentos senol\u00edticos melhoram este cen\u00e1rio inflamat\u00f3rio, eliminando as c\u00e9lulas senescentes e poupando as saud\u00e1veis.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Embora existam aproximadamente 80 senol\u00edticos conhecidos, apenas uma combina\u00e7\u00e3o de dois, dasatinib e quercetina, foi testada em humanos.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">A descoberta de medicamentos \u00e9 excecionalmente dispendiosa e demora normalmente 10 a 20 anos - \u00e9 um estrangulamento significativo na cadeia de desenvolvimento de medicamentos. Neste estudo, os investigadores utilizaram a aprendizagem autom\u00e1tica (AM) para acelerar a descoberta de novos medicamentos senol\u00edticos.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Treinaram modelos de IA em senol\u00edticos e n\u00e3o-senol\u00edticos existentes, permitindo \u00e0 IA distinguir entre eles e prever a probabilidade de mol\u00e9culas n\u00e3o encontradas serem senol\u00edticas.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Das 4340 mol\u00e9culas avaliadas, a IA assinalou 21 com uma elevada probabilidade de serem senol\u00edticas em 5 minutos.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Uma das autoras do estudo, a Dra. Vanessa Smer-Barreto, <\/span><a href=\"https:\/\/theconversation.com\/ai-finds-drugs-that-could-fight-ageing-and-age-related-diseases-208390#:~:text=The%20results%20showed%20that%20out,they%20work%20in%20the%20body.\"><span style=\"font-weight: 400;\">disse ao The Conversation<\/span><\/a><span style=\"font-weight: 400;\"> que, se fossem testados tradicionalmente num laborat\u00f3rio, seriam necess\u00e1rias 50 000 libras s\u00f3 para comprar os compostos, excluindo o custo do equipamento e da instala\u00e7\u00e3o.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Ap\u00f3s testes in vitro em c\u00e9lulas saud\u00e1veis e senescentes, 3 das 21 mol\u00e9culas, periplocina, oleandrina e Linkedin, eliminaram eficazmente as c\u00e9lulas senescentes, poupando as c\u00e9lulas normais.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Em outros testes, a oleandrina, um composto encontrado na planta oleandro, superou os senol\u00edticos mais conhecidos do seu g\u00e9nero.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">A equipa est\u00e1 agora a testar os tr\u00eas candidatos a senol\u00edticos em tecido pulmonar humano, prevendo-se que os resultados sejam conhecidos dentro de dois anos.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Nos \u00faltimos meses, a IA tem <\/span><a href=\"https:\/\/dailyai.com\/pt\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/\"><span style=\"font-weight: 400;\">antibi\u00f3ticos potenciais identificados<\/span><\/a><span style=\"font-weight: 400;\"> eficaz para matar bact\u00e9rias resistentes a medicamentos, e uma empresa de biotecnologia sediada em Hong Kong recebeu aprova\u00e7\u00e3o para iniciar ensaios cl\u00ednicos com um <\/span><a href=\"https:\/\/dailyai.com\/pt\/2023\/07\/first-ai-generated-drug-given-go-ahead-for-human-trials\/\"><span style=\"font-weight: 400;\">Medicamento descoberto pela IA<\/span><\/a><span style=\"font-weight: 400;\">.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">A capacidade da IA para efetuar an\u00e1lises complexas de mol\u00e9culas est\u00e1 a acelerar enormemente as condutas de desenvolvimento farmac\u00eautico, abrindo novas oportunidades para combater doen\u00e7as e afec\u00e7\u00f5es comuns e dif\u00edceis de tratar. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>Uma equipa internacional de investigadores da Universidade de Edimburgo e do Conselho Nacional de Investiga\u00e7\u00e3o espanhol IBBTEC-CSIC utilizou a IA para acelerar a descoberta de medicamentos anti-envelhecimento.  O seu estudo identificou 3 potenciais medicamentos senol\u00edticos capazes de desacelerar o envelhecimento e prevenir doen\u00e7as relacionadas com a idade. Estes medicamentos funcionam eliminando as c\u00e9lulas senescentes, frequentemente designadas por \"c\u00e9lulas zombie\". Estas c\u00e9lulas permanecem metabolicamente activas, mas s\u00e3o incapazes de se replicar. Embora a paragem da replica\u00e7\u00e3o celular funcione como um mecanismo de defesa para evitar a propaga\u00e7\u00e3o de danos celulares, n\u00e3o \u00e9 totalmente simples.  Esta medida de prote\u00e7\u00e3o destina-se principalmente a impedir a prolifera\u00e7\u00e3o de c\u00e9lulas que sofreram danos no ADN -<\/p>","protected":false},"author":2,"featured_media":2385,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[203,204,105,101],"class_list":["post-2384","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-biotech","tag-healthcare","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI accelerates discovery of anti-aging drugs in new study | DailyAI<\/title>\n<meta name=\"description\" content=\"An international team of researchers from the University of Edinburgh and the Spanish National Research Council IBBTEC-CSIC employed AI to accelerate the discovery of anti-aging drugs.\" 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