{"id":950,"date":"2023-05-27T14:40:15","date_gmt":"2023-05-27T14:40:15","guid":{"rendered":"https:\/\/dailyai.com\/?p=950"},"modified":"2023-06-01T09:26:45","modified_gmt":"2023-06-01T09:26:45","slug":"ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria","status":"publish","type":"post","link":"https:\/\/dailyai.com\/nb\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/","title":{"rendered":"AI oppdager nytt antibiotikum mot resistente bakterier"},"content":{"rendered":"<p><b>Menneskeheten har sakket akterut i kampen mot medisinresistente bakterier, men kunstig intelligens kan vise seg \u00e5 v\u00e6re v\u00e5rt hemmelige v\u00e5pen.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400\">Antibiotikaresistente patogener er ansvarlige for mellom <\/span><a href=\"https:\/\/www.thelancet.com\/journals\/lancet\/article\/PIIS0140-6736(21)02724-0\/fulltext\"><span style=\"font-weight: 400\">1 og 5 millioner d\u00f8dsfall<\/span><\/a><span style=\"font-weight: 400\"> per \u00e5r.\u00a0\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">F\u00e5 nye antibiotika har blitt utviklet i l\u00f8pet av det siste ti\u00e5ret, og de fleste er sm\u00e5 justeringer av eksisterende antibiotika.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Det er sv\u00e6rt arbeidskrevende \u00e5 finne nye legemidler, men en ny studie har utnyttet kunstig intelligens til \u00e5 automatisk screene tusenvis av stoffer for \u00e5 avdekke muligheter for laboratorietesting.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Den <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41589-023-01349-8.epdf?sharing_token=8HV9JdX6i-6DpHj0fv2wOtRgN0jAjWel9jnR3ZoTv0PgqDK_eQp8NcAST1F90jpq3WEGXG2Su3RGayoL_4HVm-885WktBHURHlCxulwlcvqKkHgdWqrHo6v6OktzRXc-zL4MsysGdAFnKBAI2wyymCj5gtw5qVJSvyZDrTK_wGIpI8eaOx1jqmIvwv1jdlYBYoAQi8TfYbpGh2Cfrhw5BG1rJNzyE_FFkgm1zzQdwpc%3D&amp;tracking_referrer=www.bbc.co.uk\"><span style=\"font-weight: 400\">studie<\/span><\/a><span style=\"font-weight: 400\">publisert i Nature Chemical Biology, fors\u00f8kte forskere fra MIT og McMaster University \u00e5 finne nye medisiner for \u00e5 drepe<\/span><i><span style=\"font-weight: 400\"> Acinetobacter baumannii<\/span><\/i><span style=\"font-weight: 400\">en bakterie som <\/span><a href=\"https:\/\/www.who.int\/news\/item\/27-02-2017-who-publishes-list-of-bacteria-for-which-new-antibiotics-are-urgently-needed\"><span style=\"font-weight: 400\">WHO identifiserte<\/span><\/a><span style=\"font-weight: 400\"> som en \"kritisk trussel\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">Forskerne brukte to maskinl\u00e6ringsmodeller (ML) for \u00e5 automatisere prosessen med \u00e5 finne legemidler <\/span><a href=\"https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC1978274\/\"><i><span style=\"font-weight: 400\">in silico<\/span><\/i><\/a><span style=\"font-weight: 400\">, som betyr \"i en datamaskin\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">Slik fungerte det:<\/span><\/p>\n<p><b>Innhentet oppl\u00e6ringsdata<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Forskerne eksponerte laboratoriedyrket <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\"> til rundt 7500 forskjellige kjemiske forbindelser, og overv\u00e5ket for \u00e5 se hvilke forbindelser som hemmet veksten av mikroben.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">De kjemiske strukturene til de stoffene som hemmet vekst, ble matet inn i en maskinl\u00e6ringsmodell (ML). P\u00e5 denne m\u00e5ten kunne modellen l\u00e6re seg de kjemiske egenskapene som var forbundet med veksthemming.<\/span><\/li>\n<\/ul>\n<p><b>Trente og testet modellen<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Etter at modellen var oppl\u00e6rt, brukte forskerne den til \u00e5 analysere et sett med 6680 forbindelser som modellen ikke hadde m\u00f8tt tidligere. Disse forbindelsene ble hentet fra Drug Repurposing Hub ved Broad Institute. Den valgte ut noen hundre forbindelser.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Forskerne valgte ut 240 av disse for \u00e5 teste dem eksperimentelt i laboratoriet.\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">De fokuserte p\u00e5 forbindelser med differensierte strukturer i forhold til eksisterende antibiotika, ettersom dette gj\u00f8r det mer sannsynlig at de unng\u00e5r antibiotikaresistens.\u00a0<\/span><\/li>\n<\/ul>\n<p><b>Eksperimentell laboratorietesting<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Laboratorietester reduserte listen til ni antibiotika.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Blant disse viste det seg at en forbindelse som opprinnelig ble utforsket som et potensielt diabetesmiddel, var ekstremt effektiv til \u00e5 drepe <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\">. Legemidlet ble kalt \"abaucin\".\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Det spesielle var at det ikke p\u00e5virket andre bakteriearter, inkludert <\/span><i><span style=\"font-weight: 400\">Pseudomonas aeruginosa, Staphylococcus aureus, <\/span><\/i><span style=\"font-weight: 400\">og <\/span><i><span style=\"font-weight: 400\">Enterobacteriaceae.<\/span><\/i><\/li>\n<\/ul>\n<p><span style=\"font-weight: 400\">Dr. Stokes, som jobbet med prosjektet, <\/span><a href=\"https:\/\/www.bbc.co.uk\/news\/health-65709834\"><span style=\"font-weight: 400\">fortalte BBC<\/span><\/a><span style=\"font-weight: 400\">\"Det er n\u00e5 arbeidet begynner.\"\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Antibiotikumet vil gjennomg\u00e5 en langvarig testprosedyre for \u00e5 m\u00e5le sikkerheten i mennesker, som kanskje ikke er ferdig f\u00f8r i 2030.<\/span><\/p>\n<p><span style=\"font-weight: 400\">AI gj\u00f8r det likevel raskere \u00e5 utforske nye legemidler, og hjelper forskerne med \u00e5 finne interessante og nye antimikrobielle forbindelser. Mange av dem har blitt utviklet til andre form\u00e5l, s\u00e5 de finnes allerede der ute - vi trenger bare \u00e5 finne dem.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Dr. Stokes sa: \"Kunstig intelligens \u00f8ker hastigheten, og i en perfekt verden reduserer kostnadene, som vi kan bruke til \u00e5 oppdage disse nye antibiotikaklassene som vi s\u00e5rt trenger.\"\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Selv om det fortsatt tar lang tid \u00e5 teste sikkerheten p\u00e5 mennesker, vil AI-st\u00f8ttede forskningspipelines helt sikkert bidra til at antibiotika og andre legemidler kommer raskere p\u00e5 markedet. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>Menneskeheten har sakket akterut i kampen mot medisinresistente bakterier, men kunstig intelligens kan vise seg \u00e5 v\u00e6re v\u00e5rt hemmelige v\u00e5pen.  Antibiotikaresistente patogener er ansvarlig for mellom 1 og 5 millioner d\u00f8dsfall per \u00e5r.   F\u00e5 nye antibiotika har blitt utviklet i l\u00f8pet av det siste ti\u00e5ret, og de fleste er sm\u00e5 justeringer av eksisterende antibiotika.  Det er sv\u00e6rt arbeidskrevende \u00e5 finne nye medisiner, men en ny studie har utnyttet kunstig intelligens til automatisk \u00e5 screene tusenvis av forbindelser for \u00e5 avdekke muligheter for laboratorietesting.  I studien, som ble publisert i Nature Chemical Biology, fors\u00f8kte forskere fra MIT og McMaster University \u00e5 finne nye legemidler som kunne drepe Acinetobacter baumannii,<\/p>","protected":false},"author":2,"featured_media":951,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[105,101],"class_list":["post-950","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI discovers new antibiotic for drug-resistant bacteria | DailyAI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" 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