{"id":2384,"date":"2023-07-07T20:16:06","date_gmt":"2023-07-07T20:16:06","guid":{"rendered":"https:\/\/dailyai.com\/?p=2384"},"modified":"2023-07-07T21:05:18","modified_gmt":"2023-07-07T21:05:18","slug":"ai-accelerates-discovery-of-anti-aging-drugs-in-new-study","status":"publish","type":"post","link":"https:\/\/dailyai.com\/it\/2023\/07\/ai-accelerates-discovery-of-anti-aging-drugs-in-new-study\/","title":{"rendered":"L'intelligenza artificiale accelera la scoperta di farmaci anti-invecchiamento in un nuovo studio"},"content":{"rendered":"<p><b>Un team internazionale di ricercatori dell'Universit\u00e0 di Edimburgo e del Consiglio Nazionale delle Ricerche spagnolo IBBTEC-CSIC ha impiegato l'intelligenza artificiale per accelerare la scoperta di farmaci anti-invecchiamento.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400;\">Il loro <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41467-023-39120-1\"><span style=\"font-weight: 400;\">studio<\/span><\/a><span style=\"font-weight: 400;\"> ha identificato 3 potenziali farmaci senolitici in grado di decelerare l'invecchiamento e prevenire le malattie legate all'et\u00e0. Questi farmaci funzionano eliminando le cellule senescenti, spesso chiamate \"cellule zombie\". Queste cellule rimangono metabolicamente attive ma non sono in grado di replicarsi.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">L'arresto della replicazione cellulare \u00e8 un meccanismo difensivo per prevenire la diffusione del danno cellulare, ma non \u00e8 del tutto semplice.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Questa misura protettiva ha lo scopo principale di impedire la proliferazione delle cellule che hanno subito danni al DNA, ad esempio quelle danneggiate dall'esposizione alla luce solare. Bloccando la replicazione di queste cellule danneggiate, l'organismo si assicura che il danno non si diffonda ad altre cellule.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Tuttavia, queste cellule che hanno smesso di dividersi, note come cellule senescenti, possono potenzialmente causare danni. Quando entrano nella fase di senescenza, iniziano a rilasciare proteine note per causare infiammazioni.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Ci\u00f2 pu\u00f2 influire sulle cellule sane vicine, creando potenzialmente un ambiente infiammatorio.\u00a0<\/span><span style=\"font-weight: 400;\">Nel tempo, questo accumulo di infiammazione pu\u00f2 contribuire a varie complicazioni di salute.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Ad esempio, l'infiammazione \u00e8 legata a molte malattie, tra cui quelle neurologiche e degenerative, il diabete di tipo 2, la fibrosi polmonare, l'osteoartrite e il cancro.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Pertanto, se da un lato l'interruzione della replicazione cellulare \u00e8 fondamentale per prevenire la diffusione del danno al DNA, dall'altro la risposta infiammatoria associata alle cellule senescenti pu\u00f2 portare ad altri problemi di salute se non viene gestita correttamente.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Ed \u00e8 qui che i farmaci senolitici possono aiutare.\u00a0<\/span><\/p>\n<h2><span style=\"font-weight: 400;\">Il ruolo dell'intelligenza artificiale<\/span><\/h2>\n<p><span style=\"font-weight: 400;\">Precedenti ricerche su topi di laboratorio hanno dimostrato che i farmaci senolitici migliorano questo scenario infiammatorio eliminando le cellule senescenti e risparmiando quelle sane.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Sebbene esistano circa 80 senolitici noti, solo una combinazione di due, dasatinib e quercetina, \u00e8 stata testata nell'uomo.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">La scoperta di farmaci \u00e8 eccezionalmente costosa e di solito richiede dai 10 ai 20 anni: \u00e8 un collo di bottiglia significativo nella pipeline di sviluppo dei farmaci. In questo studio, i ricercatori hanno utilizzato l'apprendimento automatico (ML) per accelerare la scoperta di nuovi farmaci senolitici.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Hanno addestrato modelli di intelligenza artificiale su senolitici e non senolitici esistenti, consentendo all'intelligenza artificiale di distinguerli e di prevedere la probabilit\u00e0 che le molecole non incontrate siano senolitiche.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Su 4.340 molecole valutate, l'IA ne ha segnalate 21 con un'alta probabilit\u00e0 di essere senolitiche entro 5 minuti.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Una delle autrici dello studio, la dott.ssa Vanessa Smer-Barreto, <\/span><a href=\"https:\/\/theconversation.com\/ai-finds-drugs-that-could-fight-ageing-and-age-related-diseases-208390#:~:text=The%20results%20showed%20that%20out,they%20work%20in%20the%20body.\"><span style=\"font-weight: 400;\">ha dichiarato a The Conversation<\/span><\/a><span style=\"font-weight: 400;\"> che, se testato tradizionalmente in laboratorio, richiederebbe 50.000 sterline solo per l'acquisto dei composti, escludendo il costo delle attrezzature e dell'allestimento.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">In seguito a test in vitro su cellule sane e senescenti, 3 delle 21 molecole, periplocina, oleandrina e Linkedin, hanno eliminato efficacemente le cellule senescenti risparmiando quelle normali.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">In ulteriori test, l'oleandrina, un composto presente nella pianta di oleandro, ha superato i pi\u00f9 noti senolitici di questo tipo.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Il team sta ora testando i 3 candidati senolitici su tessuto polmonare umano, con risultati attesi tra circa due anni.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Negli ultimi due mesi, l'intelligenza artificiale ha <\/span><a href=\"https:\/\/dailyai.com\/it\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/\"><span style=\"font-weight: 400;\">potenziali antibiotici identificati<\/span><\/a><span style=\"font-weight: 400;\"> efficace nell'uccidere i batteri resistenti ai farmaci, e un'azienda biotecnologica con sede a Hong Kong ha ricevuto l'approvazione per l'avvio di studi clinici con un farmaco <\/span><a href=\"https:\/\/dailyai.com\/it\/2023\/07\/first-ai-generated-drug-given-go-ahead-for-human-trials\/\"><span style=\"font-weight: 400;\">Farmaco scoperto dall'intelligenza artificiale<\/span><\/a><span style=\"font-weight: 400;\">.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">La capacit\u00e0 dell'intelligenza artificiale di eseguire analisi complesse delle molecole sta accelerando notevolmente le pipeline di sviluppo farmaceutico, aprendo nuove opportunit\u00e0 per affrontare condizioni e malattie comuni e difficili da trattare. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>Un team internazionale di ricercatori dell'Universit\u00e0 di Edimburgo e del Consiglio Nazionale delle Ricerche spagnolo IBBTEC-CSIC ha impiegato l'intelligenza artificiale per accelerare la scoperta di farmaci anti-invecchiamento.  Il loro studio ha identificato 3 potenziali farmaci senolitici in grado di decelerare l'invecchiamento e prevenire le malattie legate all'et\u00e0. Questi farmaci funzionano eliminando le cellule senescenti, spesso chiamate \"cellule zombie\". Queste cellule rimangono metabolicamente attive ma non sono in grado di replicarsi. Sebbene l'interruzione della replicazione cellulare agisca come meccanismo difensivo per prevenire la diffusione del danno cellulare, non \u00e8 del tutto semplice.  Questa misura protettiva \u00e8 pensata principalmente per impedire la proliferazione delle cellule che hanno subito un danno al DNA.<\/p>","protected":false},"author":2,"featured_media":2385,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[203,204,105,101],"class_list":["post-2384","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-biotech","tag-healthcare","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI accelerates discovery of anti-aging drugs in new study | DailyAI<\/title>\n<meta name=\"description\" content=\"An international team of researchers from the University of Edinburgh and the Spanish National Research Council IBBTEC-CSIC employed AI to accelerate the discovery of anti-aging drugs.\" 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