{"id":11639,"date":"2024-04-17T11:21:32","date_gmt":"2024-04-17T11:21:32","guid":{"rendered":"https:\/\/dailyai.com\/?p=11639"},"modified":"2024-04-17T12:42:25","modified_gmt":"2024-04-17T12:42:25","slug":"scientists-accelerate-search-for-parkinsons-treatments-using-ai","status":"publish","type":"post","link":"https:\/\/dailyai.com\/it\/2024\/04\/scientists-accelerate-search-for-parkinsons-treatments-using-ai\/","title":{"rendered":"Gli scienziati accelerano la ricerca di trattamenti per il Parkinson utilizzando l'intelligenza artificiale"},"content":{"rendered":"<p><b>I ricercatori dell'Universit\u00e0 di Cambridge hanno sfruttato l'intelligenza artificiale per accelerare drasticamente la ricerca di nuove terapie per il morbo di Parkinson.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400;\">Utilizzando tecniche di apprendimento automatico, sono stati in grado di vagliare milioni di potenziali composti farmacologici e di identificare i candidati pi\u00f9 promettenti dieci volte pi\u00f9 velocemente e 1000 volte pi\u00f9 economicamente rispetto ai metodi convenzionali.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">La malattia di Parkinson \u00e8 una malattia neurodegenerativa complessa e progressiva che affligge circa 6 milioni di persone in tutto il mondo. Si prevede che questa cifra triplicher\u00e0 entro il 2040. <\/span><\/p>\n<p><span style=\"font-weight: 400;\">Attualmente non esistono trattamenti in grado di rallentare o arrestare in modo affidabile la progressione della malattia.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Il processo tradizionale di screening di vaste librerie chimiche per trovare potenziali candidati farmaci \u00e8 estremamente lento, costoso e spesso infruttuoso.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">\"Una strada per la ricerca di potenziali trattamenti per il Parkinson richiede l'identificazione di piccole molecole in grado di inibire l'aggregazione dell'alfa-sinucleina, una proteina strettamente associata alla malattia\", ha spiegato il ricercatore principale, il professor Michele Vendruscolo. <\/span><a href=\"https:\/\/www.cam.ac.uk\/research\/news\/ai-speeds-up-drug-design-for-parkinsons-ten-fold\" target=\"_blank\" rel=\"noopener\"><span style=\"font-weight: 400;\">ha dichiarato all'Universit\u00e0 di Cambridge.<\/span><\/a><\/p>\n<p><span style=\"font-weight: 400;\">\"Ma si tratta di un processo che richiede molto tempo: la sola identificazione di un candidato principale per ulteriori test pu\u00f2 richiedere mesi o addirittura anni\".<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Per affrontare questa sfida, Vendruscolo e il suo team hanno sviluppato un approccio di apprendimento automatico in 5 fasi. Il <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41589-024-01580-x\" target=\"_blank\" rel=\"noopener\"><span style=\"font-weight: 400;\">studio<\/span><\/a><span style=\"font-weight: 400;\"> \u00e8 stato pubblicato in <em>Natura Biologia Chimica<\/em>.\u00a0<\/span><\/p>\n<ol>\n<li style=\"font-weight: 400;\" aria-level=\"1\"><span style=\"font-weight: 400;\">Iniziare con una piccola serie di composti, identificati tramite simulazioni, che mostrano il potenziale per bloccare l'aggregazione della proteina alfa-sinucleina, che \u00e8 la causa principale del Parkinson. Poi, testate sperimentalmente la loro efficacia.<\/span><\/li>\n<li style=\"font-weight: 400;\" aria-level=\"1\"><span style=\"font-weight: 400;\">Utilizzare i risultati per addestrare un modello di apprendimento automatico per prevedere quali strutture e propriet\u00e0 molecolari rendono un composto efficace nel prevenire l'aggregazione proteica.<\/span><\/li>\n<li style=\"font-weight: 400;\" aria-level=\"1\"><span style=\"font-weight: 400;\">Il modello addestrato viene utilizzato per esaminare rapidamente una libreria virtuale contenente milioni di composti e prevedere i concorrenti pi\u00f9 potenti.<\/span><\/li>\n<li style=\"font-weight: 400;\" aria-level=\"1\"><span style=\"font-weight: 400;\">Convalidare sperimentalmente in laboratorio i migliori candidati selezionati dall'AI. Alimentare questi risultati nel modello per perfezionare ulteriormente le sue capacit\u00e0 di previsione.<\/span><\/li>\n<li style=\"font-weight: 400;\" aria-level=\"1\"><span style=\"font-weight: 400;\">Ripetere questo ciclo di previsioni computazionali e test sperimentali, con il modello AI che diventa pi\u00f9 intelligente a ogni tornata, individuando i composti pi\u00f9 potenti.<\/span><\/li>\n<\/ol>\n<figure id=\"attachment_11640\" aria-describedby=\"caption-attachment-11640\" style=\"width: 685px\" class=\"wp-caption aligncenter\"><img loading=\"lazy\" decoding=\"async\" class=\"wp-image-11640 size-full\" src=\"https:\/\/dailyai.com\/wp-content\/uploads\/2024\/04\/41589_2024_1580_Figa_HTML.webp\" alt=\"AI Parkinson\" width=\"685\" height=\"395\" srcset=\"https:\/\/dailyai.com\/wp-content\/uploads\/2024\/04\/41589_2024_1580_Figa_HTML.webp 685w, https:\/\/dailyai.com\/wp-content\/uploads\/2024\/04\/41589_2024_1580_Figa_HTML-300x173.webp 300w, https:\/\/dailyai.com\/wp-content\/uploads\/2024\/04\/41589_2024_1580_Figa_HTML-60x35.webp 60w\" sizes=\"auto, (max-width: 685px) 100vw, 685px\" \/><figcaption id=\"caption-attachment-11640\" class=\"wp-caption-text\">Il sistema iterativo dell'Universit\u00e0 di Cambridge per la scoperta di farmaci contro il Parkinson. Fonte: <a href=\"https:\/\/www.nature.com\/articles\/s41589-024-01580-x\">Natura Biologia Chimica<\/a> (accesso libero)<\/figcaption><\/figure>\n<p><span style=\"font-weight: 400;\">Nel corso di pi\u00f9 iterazioni, il tasso di ottimizzazione - la percentuale di composti testati che inibiscono l'aggregazione di alfa-sinucleina associata al Parkinson - \u00e8 aumentato da 4% a oltre 20%.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Inoltre, i composti trovati dall'IA erano, in media, molto pi\u00f9 potenti di quelli precedentemente identificati. Alcuni hanno mostrato un'attivit\u00e0 promettente a dosi otto volte inferiori. Erano anche pi\u00f9 diversificati dal punto di vista chimico: il modello ha scoperto composti efficaci che differivano dalle strutture note.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">\"L'apprendimento automatico sta avendo un impatto reale sulla scoperta dei farmaci, accelerando l'intero processo di identificazione dei candidati pi\u00f9 promettenti\", ha dichiarato Vendruscolo. <\/span><\/p>\n<p><span style=\"font-weight: 400;\">\"Utilizzando le conoscenze acquisite dallo screening iniziale con il nostro modello di apprendimento automatico, siamo stati in grado di addestrare il modello per identificare le regioni specifiche di queste piccole molecole responsabili del legame, in modo da poter effettuare un nuovo screening e trovare molecole pi\u00f9 potenti.\"<\/span><\/p>\n<p><span style=\"font-weight: 400;\">\"Per noi questo significa poter iniziare a lavorare su pi\u00f9 programmi di scoperta di farmaci, invece che su uno solo. Grazie alla massiccia riduzione dei tempi e dei costi, \u00e8 possibile fare molto: \u00e8 un momento entusiasmante\".<\/span><\/p>\n<p><span style=\"font-weight: 400;\">I ricercatori sottolineano che questo \u00e8 solo l'inizio di ci\u00f2 che gli approcci AI potrebbero consentire nella scoperta di farmaci per il Parkinson e altre malattie caratterizzate da misfolding e aggregazione delle proteine.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Con l'ulteriore sviluppo e con set di dati di addestramento pi\u00f9 ampi, il potere predittivo di questi modelli non potr\u00e0 che migliorare.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Sebbene la strada da percorrere per trasformare questi candidati identificati dall'intelligenza artificiale in trattamenti approvati sia ancora lunga, questo studio dimostra come l'apprendimento automatico, abilmente combinato con la biologia sperimentale, possa accelerare notevolmente le prime fasi della scoperta di farmaci.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Questo si basa su una serie di ricerche che affrontano la sfida della ricerca di nuovi trattamenti farmacologici, tra cui <\/span><a href=\"https:\/\/dailyai.com\/it\/2023\/06\/researchers-build-breakthrough-ai-model-for-drug-discovery\/\"><span style=\"font-weight: 400;\">dal MIT e da Tufts<\/span><\/a><span style=\"font-weight: 400;\">che ha recentemente costruito un modello in grado di vagliare circa 100 milioni di composti al giorno. <\/span><\/p>\n<p><span style=\"font-weight: 400;\">Diversi <\/span><a href=\"https:\/\/dailyai.com\/it\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/\"><span style=\"font-weight: 400;\">modelli di scoperta degli antibiotici<\/span><\/a><span style=\"font-weight: 400;\"> hanno prodotto composti sperimentali, alcuni dei quali sono <a href=\"https:\/\/dailyai.com\/it\/2023\/07\/first-ai-generated-drug-given-go-ahead-for-human-trials\/\">verso le sperimentazioni cliniche<\/a>.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Un altro <\/span><a href=\"https:\/\/dailyai.com\/it\/2023\/08\/ai-eye-scan-yields-excellent-results-for-parkinsons-disease-early-detection\/\"><span style=\"font-weight: 400;\">progetto su larga scala<\/span><\/a><span style=\"font-weight: 400;\"> in collaborazione con il Moorfields Eye Hospital nel Regno Unito, l'anno scorso ha utilizzato le scansioni oculari per identificare i primi segni del Parkinson - un metodo innovativo abilitato dall'intelligenza artificiale.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Con questo nuovo studio che mira a scoprire trattamenti efficaci per il Parkinson, i metodi di intelligenza artificiale mostrano un'immensa promessa di ridefinizione della medicina e dell'assistenza sanitaria.\u00a0<\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>I ricercatori dell'Universit\u00e0 di Cambridge hanno sfruttato l'intelligenza artificiale per accelerare drasticamente la ricerca di nuove terapie per il morbo di Parkinson.  Utilizzando tecniche di apprendimento automatico, sono stati in grado di vagliare milioni di potenziali composti farmacologici e di identificare i candidati pi\u00f9 promettenti dieci volte pi\u00f9 velocemente e 1000 volte pi\u00f9 economicamente rispetto ai metodi convenzionali. Il morbo di Parkinson \u00e8 una malattia neurodegenerativa complessa e progressiva che affligge circa 6 milioni di persone in tutto il mondo. Si prevede che questa cifra triplicher\u00e0 entro il 2040. Attualmente, nessun trattamento \u00e8 in grado di rallentare o arrestare in modo affidabile la progressione della malattia.  Il processo tradizionale di screening di vaste biblioteche chimiche per trovare potenziali candidati farmaci \u00e8 estremamente<\/p>","protected":false},"author":2,"featured_media":11641,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[204,178],"class_list":["post-11639","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-healthcare","tag-medicine"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.3 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Scientists accelerate the search for Parkinson&#039;s treatments using AI | DailyAI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/dailyai.com\/it\/2024\/04\/scientists-accelerate-search-for-parkinsons-treatments-using-ai\/\" \/>\n<meta property=\"og:locale\" content=\"it_IT\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Scientists accelerate the search for Parkinson&#039;s treatments using AI | DailyAI\" \/>\n<meta property=\"og:description\" content=\"Researchers at the University of Cambridge have harnessed AI to dramatically accelerate the search for new Parkinson&#8217;s disease therapies.\u00a0 By using machine learning techniques, they were able to screen millions of potential drug compounds and identify the most promising candidates ten times faster and 1000 times more cost-effectively than conventional methods. Parkinson&#8217;s disease is a complex, progressive neurodegenerative disease that afflicts approximately 6 million people worldwide. That figure is expected to triple by 2040. Currently, no treatments can reliably slow or halt the disease&#8217;s progression.\u00a0 The traditional process of screening vast chemical libraries to find potential drug candidates is extremely\" \/>\n<meta property=\"og:url\" content=\"https:\/\/dailyai.com\/it\/2024\/04\/scientists-accelerate-search-for-parkinsons-treatments-using-ai\/\" \/>\n<meta property=\"og:site_name\" content=\"DailyAI\" \/>\n<meta property=\"article:published_time\" content=\"2024-04-17T11:21:32+00:00\" \/>\n<meta property=\"article:modified_time\" content=\"2024-04-17T12:42:25+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/dailyai.com\/wp-content\/uploads\/2024\/04\/DALL\u00b7E-2024-04-17-12.16.35-A-modern-high-tech-laboratory-specifically-focused-on-Parkinsons-disease-research-but-without-any-people.-The-scene-includes-sleek-futuristic-devi.webp\" \/>\n\t<meta property=\"og:image:width\" content=\"1792\" \/>\n\t<meta property=\"og:image:height\" content=\"1024\" \/>\n\t<meta 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