{"id":950,"date":"2023-05-27T14:40:15","date_gmt":"2023-05-27T14:40:15","guid":{"rendered":"https:\/\/dailyai.com\/?p=950"},"modified":"2023-06-01T09:26:45","modified_gmt":"2023-06-01T09:26:45","slug":"ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria","status":"publish","type":"post","link":"https:\/\/dailyai.com\/es\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/","title":{"rendered":"La IA descubre un nuevo antibi\u00f3tico contra las bacterias resistentes a los medicamentos"},"content":{"rendered":"<p><b>La humanidad se ha quedado atr\u00e1s en la lucha contra las bacterias resistentes a los medicamentos, pero la IA podr\u00eda ser nuestra arma secreta.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400\">Los pat\u00f3genos resistentes a los antibi\u00f3ticos son responsables de entre <\/span><a href=\"https:\/\/www.thelancet.com\/journals\/lancet\/article\/PIIS0140-6736(21)02724-0\/fulltext\"><span style=\"font-weight: 400\">1 y 5 millones de muertes<\/span><\/a><span style=\"font-weight: 400\"> al a\u00f1o.\u00a0\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">En la \u00faltima d\u00e9cada se han desarrollado pocos antibi\u00f3ticos nuevos, y la mayor\u00eda son ligeros retoques de los ya existentes.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Descubrir nuevos f\u00e1rmacos es una tarea excepcionalmente laboriosa, pero un estudio reciente ha aprovechado la inteligencia artificial para examinar autom\u00e1ticamente miles de compuestos y descubrir v\u00edas de ensayo en laboratorio.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">En <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41589-023-01349-8.epdf?sharing_token=8HV9JdX6i-6DpHj0fv2wOtRgN0jAjWel9jnR3ZoTv0PgqDK_eQp8NcAST1F90jpq3WEGXG2Su3RGayoL_4HVm-885WktBHURHlCxulwlcvqKkHgdWqrHo6v6OktzRXc-zL4MsysGdAFnKBAI2wyymCj5gtw5qVJSvyZDrTK_wGIpI8eaOx1jqmIvwv1jdlYBYoAQi8TfYbpGh2Cfrhw5BG1rJNzyE_FFkgm1zzQdwpc%3D&amp;tracking_referrer=www.bbc.co.uk\"><span style=\"font-weight: 400\">estudiar<\/span><\/a><span style=\"font-weight: 400\">publicado en Nature Chemical Biology, investigadores del MIT y de la Universidad McMaster intentan descubrir nuevos f\u00e1rmacos que maten a los animales.<\/span><i><span style=\"font-weight: 400\"> Acinetobacter baumannii<\/span><\/i><span style=\"font-weight: 400\">una bacteria que la <\/span><a href=\"https:\/\/www.who.int\/news\/item\/27-02-2017-who-publishes-list-of-bacteria-for-which-new-antibiotics-are-urgently-needed\"><span style=\"font-weight: 400\">La OMS identific\u00f3<\/span><\/a><span style=\"font-weight: 400\"> como una \"amenaza cr\u00edtica\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">Los investigadores utilizaron dos modelos de aprendizaje autom\u00e1tico (ML) para automatizar el proceso de descubrimiento de f\u00e1rmacos <\/span><a href=\"https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC1978274\/\"><i><span style=\"font-weight: 400\">in silico<\/span><\/i><\/a><span style=\"font-weight: 400\">que significa \"en un ordenador\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">Funcionaba as\u00ed:<\/span><\/p>\n<p><b>Datos de entrenamiento obtenidos<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Los investigadores expusieron <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\"> a unos 7.500 compuestos qu\u00edmicos diferentes y se control\u00f3 qu\u00e9 compuestos inhib\u00edan el crecimiento del microbio.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Las estructuras qu\u00edmicas de los inhibidores del crecimiento se introdujeron en un modelo de aprendizaje autom\u00e1tico. Esto permiti\u00f3 al modelo aprender las caracter\u00edsticas qu\u00edmicas asociadas a la inhibici\u00f3n del crecimiento.<\/span><\/li>\n<\/ul>\n<p><b>Entrenamiento y prueba del modelo<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Una vez entrenado el modelo, los investigadores lo utilizaron para analizar un conjunto de 6.680 compuestos que el modelo no hab\u00eda encontrado antes. Estos compuestos proced\u00edan del Drug Repurposing Hub del Broad Institute. Se seleccionaron unos cientos de compuestos.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Los investigadores eligieron 240 de la lista para realizar pruebas experimentales en el laboratorio.\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Se centraron en compuestos con estructuras diferenciadas de los antibi\u00f3ticos existentes, ya que as\u00ed es m\u00e1s probable que eludan la resistencia a los antibi\u00f3ticos.\u00a0<\/span><\/li>\n<\/ul>\n<p><b>Pruebas experimentales de laboratorio<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Las pruebas de laboratorio redujeron la lista a 9 antibi\u00f3ticos.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Entre ellos, un compuesto estudiado inicialmente como posible f\u00e1rmaco contra la diabetes result\u00f3 ser extremadamente eficaz para matar <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\">. El medicamento se llamaba \"abaucina\".\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Curiosamente, no afect\u00f3 a otras especies de bacterias, entre ellas <\/span><i><span style=\"font-weight: 400\">Pseudomonas aeruginosa, Staphylococcus aureus, <\/span><\/i><span style=\"font-weight: 400\">y <\/span><i><span style=\"font-weight: 400\">Enterobacteriaceae.<\/span><\/i><\/li>\n<\/ul>\n<p><span style=\"font-weight: 400\">Dr. Stokes, que trabaj\u00f3 en el proyecto, <\/span><a href=\"https:\/\/www.bbc.co.uk\/news\/health-65709834\"><span style=\"font-weight: 400\">a la BBC<\/span><\/a><span style=\"font-weight: 400\">\"Ahora es cuando empieza el trabajo\".\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">El antibi\u00f3tico se someter\u00e1 a un largo proceso de pruebas para evaluar su seguridad en humanos, que podr\u00eda no concluir hasta 2030.<\/span><\/p>\n<p><span style=\"font-weight: 400\">Aun as\u00ed, la IA acelera la laboriosa tarea de explorar nuevos f\u00e1rmacos, ayudando a los investigadores a descubrir compuestos antimicrobianos interesantes y novedosos. Muchos se han desarrollado para otros fines, as\u00ed que ya est\u00e1n ah\u00ed fuera, solo hay que encontrarlos.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Seg\u00fan el Dr. Stokes, \"la IA aumenta el ritmo, y en un mundo perfecto disminuye el coste, con el que podemos descubrir estas nuevas clases de antibi\u00f3ticos que necesitamos desesperadamente.\"\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Aunque las pruebas de seguridad en humanos siguen siendo un proceso lento, las l\u00edneas de investigaci\u00f3n basadas en IA acelerar\u00e1n sin duda la comercializaci\u00f3n de antibi\u00f3ticos y otros f\u00e1rmacos. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>La humanidad se ha quedado atr\u00e1s en la lucha contra las bacterias resistentes a los medicamentos, pero la IA podr\u00eda ser nuestra arma secreta.  Los pat\u00f3genos resistentes a los antibi\u00f3ticos son responsables de entre 1 y 5 millones de muertes al a\u00f1o.   En la \u00faltima d\u00e9cada se han desarrollado pocos antibi\u00f3ticos nuevos, y la mayor\u00eda son ligeros retoques de los ya existentes.  Descubrir nuevos f\u00e1rmacos requiere mucho trabajo, pero un estudio reciente ha aprovechado la inteligencia artificial para analizar autom\u00e1ticamente miles de compuestos y descubrir v\u00edas de ensayo en laboratorio.  En el estudio, publicado en Nature Chemical Biology, investigadores del MIT y de la Universidad McMaster intentaron descubrir nuevos f\u00e1rmacos contra la bacteria Acinetobacter baumannii,<\/p>","protected":false},"author":2,"featured_media":951,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[105,101],"class_list":["post-950","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI discovers new antibiotic for drug-resistant bacteria | DailyAI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" 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