{"id":2384,"date":"2023-07-07T20:16:06","date_gmt":"2023-07-07T20:16:06","guid":{"rendered":"https:\/\/dailyai.com\/?p=2384"},"modified":"2023-07-07T21:05:18","modified_gmt":"2023-07-07T21:05:18","slug":"ai-accelerates-discovery-of-anti-aging-drugs-in-new-study","status":"publish","type":"post","link":"https:\/\/dailyai.com\/es\/2023\/07\/ai-accelerates-discovery-of-anti-aging-drugs-in-new-study\/","title":{"rendered":"La IA acelera el descubrimiento de f\u00e1rmacos antienvejecimiento en un nuevo estudio"},"content":{"rendered":"<p><b>Un equipo internacional de investigadores de la Universidad de Edimburgo y el Consejo Superior de Investigaciones Cient\u00edficas IBBTEC-CSIC emple\u00f3 la IA para acelerar el descubrimiento de f\u00e1rmacos contra el envejecimiento.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400;\">Su <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41467-023-39120-1\"><span style=\"font-weight: 400;\">estudiar<\/span><\/a><span style=\"font-weight: 400;\"> identificaron 3 posibles f\u00e1rmacos senol\u00edticos capaces de desacelerar el envejecimiento y prevenir las enfermedades relacionadas con la edad. Estos f\u00e1rmacos act\u00faan eliminando las c\u00e9lulas senescentes, a menudo denominadas \"c\u00e9lulas zombi\". Estas c\u00e9lulas permanecen metab\u00f3licamente activas pero son incapaces de replicarse.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Aunque detener la replicaci\u00f3n celular act\u00faa como mecanismo defensivo para evitar la propagaci\u00f3n del da\u00f1o celular, no es del todo sencillo.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Esta medida protectora est\u00e1 dise\u00f1ada principalmente para evitar la proliferaci\u00f3n de c\u00e9lulas que han sufrido da\u00f1os en el ADN, por ejemplo, c\u00e9lulas da\u00f1adas por la exposici\u00f3n a la luz solar. Al detener la replicaci\u00f3n de estas c\u00e9lulas da\u00f1adas, el organismo se asegura de que este da\u00f1o no se propague a m\u00e1s c\u00e9lulas.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Sin embargo, estas c\u00e9lulas que han dejado de dividirse, conocidas como c\u00e9lulas senescentes, pueden potencialmente causar da\u00f1os. Cuando entran en la fase de senescencia, empiezan a liberar prote\u00ednas conocidas por causar inflamaci\u00f3n.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Esto puede afectar a las c\u00e9lulas sanas vecinas, creando potencialmente un entorno inflamatorio.\u00a0<\/span><span style=\"font-weight: 400;\">Con el tiempo, esta acumulaci\u00f3n de inflamaci\u00f3n puede contribuir a diversas complicaciones de salud.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Por ejemplo, la inflamaci\u00f3n est\u00e1 relacionada con muchas enfermedades, como las neurol\u00f3gicas y degenerativas, la diabetes de tipo 2, la fibrosis pulmonar, la artrosis y el c\u00e1ncer.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Por lo tanto, aunque el cese de la replicaci\u00f3n celular es crucial para prevenir la propagaci\u00f3n de da\u00f1os en el ADN, la respuesta inflamatoria asociada a las c\u00e9lulas senescentes puede provocar otros problemas de salud si no se trata adecuadamente.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Y ah\u00ed es donde los f\u00e1rmacos senol\u00edticos pueden ayudar.\u00a0<\/span><\/p>\n<h2><span style=\"font-weight: 400;\">El papel de la IA<\/span><\/h2>\n<p><span style=\"font-weight: 400;\">Investigaciones anteriores en ratones de laboratorio demostraron que los f\u00e1rmacos senol\u00edticos mejoran este escenario inflamatorio al eliminar las c\u00e9lulas senescentes y preservar las sanas.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Aunque existen aproximadamente 80 senol\u00edticos conocidos, s\u00f3lo se ha probado en humanos una combinaci\u00f3n de dos, dasatinib y quercetina.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">El descubrimiento de f\u00e1rmacos es excepcionalmente costoso y suele llevar entre 10 y 20 a\u00f1os, lo que supone un importante cuello de botella en el proceso de desarrollo de medicamentos. En este estudio, los investigadores utilizaron el aprendizaje autom\u00e1tico para acelerar el descubrimiento de nuevos f\u00e1rmacos senol\u00edticos.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Entrenaron modelos de IA con senol\u00edticos y no senol\u00edticos existentes, lo que permiti\u00f3 a la IA discernir entre ellos y predecir la probabilidad de que mol\u00e9culas no encontradas fueran senol\u00edticas.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">De 4.340 mol\u00e9culas evaluadas, la IA marc\u00f3 21 con una alta probabilidad de ser senol\u00edticas en 5 minutos.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Una de las autoras del estudio, la Dra. Vanessa Smer-Barreto, <\/span><a href=\"https:\/\/theconversation.com\/ai-finds-drugs-that-could-fight-ageing-and-age-related-diseases-208390#:~:text=The%20results%20showed%20that%20out,they%20work%20in%20the%20body.\"><span style=\"font-weight: 400;\">a The Conversation<\/span><\/a><span style=\"font-weight: 400;\"> que, si se probaran de forma tradicional en un laboratorio, se necesitar\u00edan 50.000 libras s\u00f3lo para comprar los compuestos, sin contar el coste del equipo y la instalaci\u00f3n.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Tras realizar pruebas in vitro en c\u00e9lulas sanas y senescentes, 3 de las 21 mol\u00e9culas, periplocina, oleandrina y Linkedin, eliminaron eficazmente las c\u00e9lulas senescentes y preservaron las c\u00e9lulas normales.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">En otras pruebas, la oleandrina, un compuesto de la planta de adelfa, super\u00f3 a los senol\u00edticos m\u00e1s conocidos de su clase.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">El equipo est\u00e1 probando ahora los 3 candidatos a senol\u00edticos en tejido pulmonar humano, y se esperan los resultados en unos dos a\u00f1os.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">En los \u00faltimos meses, la IA ha <\/span><a href=\"https:\/\/dailyai.com\/es\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/\"><span style=\"font-weight: 400;\">antibi\u00f3ticos potenciales identificados<\/span><\/a><span style=\"font-weight: 400;\"> eficaz para eliminar las bacterias resistentes a los medicamentos, y una empresa de biotecnolog\u00eda con sede en Hong Kong recibi\u00f3 la aprobaci\u00f3n para iniciar ensayos cl\u00ednicos con un <\/span><a href=\"https:\/\/dailyai.com\/es\/2023\/07\/first-ai-generated-drug-given-go-ahead-for-human-trials\/\"><span style=\"font-weight: 400;\">Medicamento descubierto por la IA<\/span><\/a><span style=\"font-weight: 400;\">.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">La capacidad de la IA para realizar an\u00e1lisis complejos de mol\u00e9culas est\u00e1 acelerando enormemente los procesos de desarrollo farmac\u00e9utico, abriendo nuevas oportunidades para abordar afecciones y enfermedades comunes y dif\u00edciles de tratar. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>Un equipo internacional de investigadores de la Universidad de Edimburgo y el Consejo Superior de Investigaciones Cient\u00edficas (IBBTEC-CSIC) emple\u00f3 la IA para acelerar el descubrimiento de f\u00e1rmacos antienvejecimiento.  Su estudio identific\u00f3 3 posibles f\u00e1rmacos senol\u00edticos capaces de desacelerar el envejecimiento y prevenir enfermedades relacionadas con la edad. Estos f\u00e1rmacos act\u00faan eliminando las c\u00e9lulas senescentes, a menudo denominadas \"c\u00e9lulas zombi\". Estas c\u00e9lulas permanecen metab\u00f3licamente activas pero son incapaces de replicarse. Aunque detener la replicaci\u00f3n celular act\u00faa como mecanismo defensivo para evitar la propagaci\u00f3n del da\u00f1o celular, no es del todo sencillo.  Esta medida protectora est\u00e1 dise\u00f1ada principalmente para evitar la proliferaci\u00f3n de las c\u00e9lulas que han sufrido da\u00f1os en el ADN -.<\/p>","protected":false},"author":2,"featured_media":2385,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[203,204,105,101],"class_list":["post-2384","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-biotech","tag-healthcare","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI accelerates discovery of anti-aging drugs in new study | DailyAI<\/title>\n<meta name=\"description\" content=\"An international team of researchers from the University of Edinburgh and the Spanish National Research Council IBBTEC-CSIC employed AI to accelerate the discovery of 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