{"id":2384,"date":"2023-07-07T20:16:06","date_gmt":"2023-07-07T20:16:06","guid":{"rendered":"https:\/\/dailyai.com\/?p=2384"},"modified":"2023-07-07T21:05:18","modified_gmt":"2023-07-07T21:05:18","slug":"ai-accelerates-discovery-of-anti-aging-drugs-in-new-study","status":"publish","type":"post","link":"https:\/\/dailyai.com\/de\/2023\/07\/ai-accelerates-discovery-of-anti-aging-drugs-in-new-study\/","title":{"rendered":"Neue Studie: KI beschleunigt die Entdeckung von Anti-Aging-Medikamenten"},"content":{"rendered":"<p><b>Ein internationales Forscherteam der Universit\u00e4t Edinburgh und des spanischen Nationalen Forschungsrats IBBTEC-CSIC hat KI eingesetzt, um die Entdeckung von Medikamenten gegen das Altern zu beschleunigen.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400;\">Ihre <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41467-023-39120-1\"><span style=\"font-weight: 400;\">Studie<\/span><\/a><span style=\"font-weight: 400;\"> 3 potenzielle senolytische Medikamente identifiziert, die das Altern verlangsamen und altersbedingte Krankheiten verhindern k\u00f6nnen. Diese Medikamente eliminieren seneszente Zellen, die oft als \"Zombiezellen\" bezeichnet werden. Diese Zellen bleiben metabolisch aktiv, sind aber nicht in der Lage, sich zu vermehren.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Die Unterbrechung der Zellvermehrung ist zwar ein Abwehrmechanismus, um die Ausbreitung von Zellsch\u00e4den zu verhindern, aber sie ist nicht ganz einfach.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Diese Schutzma\u00dfnahme dient in erster Linie dazu, die Vermehrung von Zellen zu verhindern, die einen DNA-Schaden erlitten haben - zum Beispiel Zellen, die durch Sonneneinstrahlung gesch\u00e4digt wurden. Indem der K\u00f6rper die Replikation dieser gesch\u00e4digten Zellen stoppt, stellt er sicher, dass sich dieser Schaden nicht auf weitere Zellen ausbreitet.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Diese Zellen, die sich nicht mehr teilen, so genannte seneszente Zellen, k\u00f6nnen jedoch potenziell Schaden anrichten. Wenn sie in die Seneszenzphase eintreten, beginnen sie, Proteine freizusetzen, die bekannterma\u00dfen Entz\u00fcndungen verursachen.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Dies kann sich auf benachbarte gesunde Zellen auswirken und m\u00f6glicherweise ein entz\u00fcndliches Umfeld schaffen.\u00a0<\/span><span style=\"font-weight: 400;\">Mit der Zeit kann diese Ansammlung von Entz\u00fcndungen zu verschiedenen gesundheitlichen Komplikationen beitragen.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">So werden Entz\u00fcndungen mit vielen Krankheiten in Verbindung gebracht, darunter neurologische und degenerative Erkrankungen, Typ-2-Diabetes, Lungenfibrose, Osteoarthritis und Krebs.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">W\u00e4hrend die Einstellung der Zellreplikation entscheidend ist, um die Ausbreitung von DNA-Sch\u00e4den zu verhindern, kann die mit alternden Zellen verbundene Entz\u00fcndungsreaktion zu anderen Gesundheitsproblemen f\u00fchren, wenn sie nicht richtig behandelt wird.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Und genau hier k\u00f6nnen senolytische Medikamente helfen.\u00a0<\/span><\/p>\n<h2><span style=\"font-weight: 400;\">Die Rolle der KI<\/span><\/h2>\n<p><span style=\"font-weight: 400;\">Fr\u00fchere Forschungen an Laborm\u00e4usen haben gezeigt, dass senolytische Medikamente dieses Entz\u00fcndungsszenario verbessern, indem sie seneszente Zellen eliminieren und gesunde Zellen verschonen.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Es gibt zwar etwa 80 bekannte Senolytika, aber nur eine Kombination von zwei, Dasatinib und Quercetin, wurde am Menschen getestet.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Die Entdeckung von Arzneimitteln ist au\u00dferordentlich kostspielig und dauert in der Regel 10 bis 20 Jahre - ein erheblicher Engpass in der Arzneimittelentwicklungspipeline. In dieser Studie setzten die Forscher maschinelles Lernen (ML) ein, um die Entdeckung neuer senolytischer Medikamente zu beschleunigen.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Sie trainierten KI-Modelle auf vorhandene Senolytika und Nicht-Senolytika, so dass die KI zwischen ihnen unterscheiden und die Wahrscheinlichkeit vorhersagen konnte, dass nicht erkannte Molek\u00fcle Senolytika sind.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Von 4.340 bewerteten Molek\u00fclen hat die KI innerhalb von 5 Minuten 21 mit hoher Wahrscheinlichkeit als senolytisch eingestuft.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Eine der Studienautorinnen, Dr. Vanessa Smer-Barreto, <\/span><a href=\"https:\/\/theconversation.com\/ai-finds-drugs-that-could-fight-ageing-and-age-related-diseases-208390#:~:text=The%20results%20showed%20that%20out,they%20work%20in%20the%20body.\"><span style=\"font-weight: 400;\">gegen\u00fcber The Conversation<\/span><\/a><span style=\"font-weight: 400;\"> dass bei herk\u00f6mmlichen Labortests allein f\u00fcr den Kauf der Pr\u00e4parate 50.000 Pfund ben\u00f6tigt w\u00fcrden, ohne die Kosten f\u00fcr Ausr\u00fcstung und Einrichtung.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Nach In-vitro-Tests an gesunden und seneszenten Zellen konnten drei der 21 Molek\u00fcle, Periplocin, Oleandrin und Linkedin, seneszente Zellen wirksam eliminieren, w\u00e4hrend normale Zellen geschont wurden.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">In weiteren Tests \u00fcbertraf Oleandrin, eine in der Oleanderpflanze enthaltene Verbindung, die bekanntesten Senolytika ihrer Art.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Das Team testet nun die drei Senolytika-Kandidaten an menschlichem Lungengewebe, wobei die Ergebnisse in etwa zwei Jahren erwartet werden.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">In den letzten Monaten hat die KI <\/span><a href=\"https:\/\/dailyai.com\/de\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/\"><span style=\"font-weight: 400;\">identifizierte potenzielle Antibiotika<\/span><\/a><span style=\"font-weight: 400;\"> wirksam bei der Abt\u00f6tung arzneimittelresistenter Bakterien, und ein in Hongkong ans\u00e4ssiges Biotech-Unternehmen erhielt die Genehmigung f\u00fcr den Beginn klinischer Versuche mit einem <\/span><a href=\"https:\/\/dailyai.com\/de\/2023\/07\/first-ai-generated-drug-given-go-ahead-for-human-trials\/\"><span style=\"font-weight: 400;\">KI-entdecktes Medikament<\/span><\/a><span style=\"font-weight: 400;\">.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Die F\u00e4higkeit der k\u00fcnstlichen Intelligenz, komplexe Molek\u00fclanalysen durchzuf\u00fchren, beschleunigt die pharmazeutischen Entwicklungspipelines erheblich und er\u00f6ffnet neue M\u00f6glichkeiten f\u00fcr die Behandlung h\u00e4ufiger und schwer zu behandelnder Krankheiten. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>Ein internationales Forscherteam von der Universit\u00e4t Edinburgh und dem spanischen Nationalen Forschungsrat IBBTEC-CSIC hat KI eingesetzt, um die Entdeckung von Medikamenten gegen das Altern zu beschleunigen.  In ihrer Studie wurden drei potenzielle senolytische Medikamente identifiziert, die das Altern verlangsamen und altersbedingte Krankheiten verhindern k\u00f6nnen. Diese Medikamente eliminieren seneszente Zellen, die oft als 'Zombie-Zellen' bezeichnet werden. Diese Zellen bleiben metabolisch aktiv, sind aber nicht in der Lage, sich zu vermehren. Die Unterbrechung der Zellreplikation ist zwar ein Schutzmechanismus, um die Ausbreitung von Zellsch\u00e4den zu verhindern, aber sie ist nicht ganz einfach.  Diese Schutzma\u00dfnahme zielt in erster Linie darauf ab, die Vermehrung von Zellen zu verhindern, die einen DNA-Schaden erlitten haben.<\/p>","protected":false},"author":2,"featured_media":2385,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[203,204,105,101],"class_list":["post-2384","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-biotech","tag-healthcare","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI accelerates discovery of anti-aging drugs in new study | DailyAI<\/title>\n<meta name=\"description\" content=\"An international team of researchers from the University of Edinburgh and the Spanish National Research Council IBBTEC-CSIC employed AI to accelerate the discovery of anti-aging drugs.\" 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