{"id":950,"date":"2023-05-27T14:40:15","date_gmt":"2023-05-27T14:40:15","guid":{"rendered":"https:\/\/dailyai.com\/?p=950"},"modified":"2023-06-01T09:26:45","modified_gmt":"2023-06-01T09:26:45","slug":"ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria","status":"publish","type":"post","link":"https:\/\/dailyai.com\/da\/2023\/05\/ai-helps-researchers-discover-a-new-antibiotic-for-treating-drug-resistant-bacteria\/","title":{"rendered":"AI opdager nyt antibiotikum til resistente bakterier"},"content":{"rendered":"<p><b>Menneskeheden er kommet bagud i kampen mod resistente bakterier, men AI kan vise sig at v\u00e6re vores hemmelige v\u00e5ben.\u00a0<\/b><\/p>\n<p><span style=\"font-weight: 400\">Antibiotikaresistente patogener er ansvarlige for mellem <\/span><a href=\"https:\/\/www.thelancet.com\/journals\/lancet\/article\/PIIS0140-6736(21)02724-0\/fulltext\"><span style=\"font-weight: 400\">1 og 5 millioner d\u00f8dsfald<\/span><\/a><span style=\"font-weight: 400\"> om \u00e5ret.\u00a0\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Der er kun udviklet f\u00e5 nye antibiotika i l\u00f8bet af det sidste \u00e5rti, og de fleste er sm\u00e5 justeringer af eksisterende antibiotika.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Det er us\u00e6dvanligt arbejdskr\u00e6vende at finde nye l\u00e6gemidler, men et nyt skels\u00e6ttende studie har udnyttet kunstig intelligens til automatisk at screene tusindvis af stoffer for at afd\u00e6kke muligheder for laboratorietest.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Den <\/span><a href=\"https:\/\/www.nature.com\/articles\/s41589-023-01349-8.epdf?sharing_token=8HV9JdX6i-6DpHj0fv2wOtRgN0jAjWel9jnR3ZoTv0PgqDK_eQp8NcAST1F90jpq3WEGXG2Su3RGayoL_4HVm-885WktBHURHlCxulwlcvqKkHgdWqrHo6v6OktzRXc-zL4MsysGdAFnKBAI2wyymCj5gtw5qVJSvyZDrTK_wGIpI8eaOx1jqmIvwv1jdlYBYoAQi8TfYbpGh2Cfrhw5BG1rJNzyE_FFkgm1zzQdwpc%3D&amp;tracking_referrer=www.bbc.co.uk\"><span style=\"font-weight: 400\">unders\u00f8gelse<\/span><\/a><span style=\"font-weight: 400\">som blev offentliggjort i Nature Chemical Biology, fors\u00f8gte forskere fra MIT og McMaster University at opdage nye l\u00e6gemidler til at dr\u00e6be<\/span><i><span style=\"font-weight: 400\"> Acinetobacter baumannii<\/span><\/i><span style=\"font-weight: 400\">en bakterie, som <\/span><a href=\"https:\/\/www.who.int\/news\/item\/27-02-2017-who-publishes-list-of-bacteria-for-which-new-antibiotics-are-urgently-needed\"><span style=\"font-weight: 400\">WHO identificerede<\/span><\/a><span style=\"font-weight: 400\"> som en \"kritisk trussel\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">Forskerne brugte to modeller for maskinl\u00e6ring (ML) til at automatisere processen for l\u00e6gemiddelopdagelse <\/span><a href=\"https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC1978274\/\"><i><span style=\"font-weight: 400\">in silico<\/span><\/i><\/a><span style=\"font-weight: 400\">som betyder \"i en computer\".<\/span><\/p>\n<p><span style=\"font-weight: 400\">S\u00e5dan her fungerede det:<\/span><\/p>\n<p><b>Indhentet tr\u00e6ningsdata<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Forskerne udsatte laboratoriedyrkede <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\"> til omkring 7.500 forskellige kemiske forbindelser og overv\u00e5get for at se, hvilke forbindelser der h\u00e6mmede mikrobens v\u00e6kst.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">De kemiske strukturer af dem, der h\u00e6mmede v\u00e6ksten, blev f\u00f8rt ind i en maskinl\u00e6ringsmodel (ML). Det gjorde det muligt for modellen at l\u00e6re de kemiske egenskaber, der er forbundet med v\u00e6ksth\u00e6mning.<\/span><\/li>\n<\/ul>\n<p><b>Tr\u00e6nede og testede modellen<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Da modellen var tr\u00e6net, brugte forskerne den til at analysere et s\u00e6t p\u00e5 6.680 forbindelser, som modellen ikke tidligere havde m\u00f8dt. Disse stoffer blev hentet fra Drug Repurposing Hub p\u00e5 Broad Institute. Den udpegede et par hundrede forbindelser.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Forskerne valgte 240 fra den korte liste til at teste eksperimentelt i laboratoriet.\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">De fokuserede p\u00e5 forbindelser med forskellige strukturer i forhold til eksisterende antibiotika, da det g\u00f8r dem mere tilb\u00f8jelige til at undg\u00e5 antibiotikaresistens.\u00a0<\/span><\/li>\n<\/ul>\n<p><b>Eksperimentel laboratorietestning<\/b><\/p>\n<ul>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Laboratorietest indsn\u00e6vrede listen til 9 antibiotika.<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">Blandt disse viste et stof, der oprindeligt blev udforsket som et potentielt diabetesmiddel, sig at v\u00e6re ekstremt effektivt til at dr\u00e6be <\/span><i><span style=\"font-weight: 400\">A. baumannii<\/span><\/i><span style=\"font-weight: 400\">. L\u00e6gemidlet blev kaldt \"abaucin\".\u00a0<\/span><\/li>\n<li style=\"font-weight: 400\"><span style=\"font-weight: 400\">M\u00e6rkeligt nok p\u00e5virkede det ikke andre bakteriearter, herunder <\/span><i><span style=\"font-weight: 400\">Pseudomonas aeruginosa, Staphylococcus aureus, <\/span><\/i><span style=\"font-weight: 400\">og <\/span><i><span style=\"font-weight: 400\">Enterobacteriaceae.<\/span><\/i><\/li>\n<\/ul>\n<p><span style=\"font-weight: 400\">Dr. Stokes, som arbejdede p\u00e5 projektet, <\/span><a href=\"https:\/\/www.bbc.co.uk\/news\/health-65709834\"><span style=\"font-weight: 400\">fortalte BBC<\/span><\/a><span style=\"font-weight: 400\">\"Det er nu, arbejdet begynder.\"\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Antibiotikummet vil gennemg\u00e5 en langvarig testprocedure for at vurdere dets sikkerhed i mennesker, som m\u00e5ske f\u00f8rst er afsluttet i 2030.<\/span><\/p>\n<p><span style=\"font-weight: 400\">Alligevel fremskynder AI den arbejdskr\u00e6vende opgave med at udforske nye l\u00e6gemidler og hj\u00e6lper forskere med at afd\u00e6kke interessante og nye antimikrobielle forbindelser. Mange af dem er blevet udviklet til andre form\u00e5l, s\u00e5 de findes allerede derude - vi skal bare finde dem.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Dr. Stokes sagde: \"AI \u00f8ger hastigheden, og i en perfekt verden reducerer det omkostningerne, hvormed vi kan opdage disse nye klasser af antibiotika, som vi desperat har brug for.\"\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400\">Selv om det stadig er en langsommelig proces at teste sikkerheden hos mennesker, vil AI-st\u00f8ttede forskningspipelines helt sikkert fremskynde time-to-market for antibiotika og andre l\u00e6gemidler. <\/span><\/p>","protected":false},"excerpt":{"rendered":"<p>Menneskeheden er kommet bagud i kampen mod medicinresistente bakterier, men AI kan vise sig at v\u00e6re vores hemmelige v\u00e5ben.  Antibiotikaresistente patogener er ansvarlige for mellem 1 og 5 millioner d\u00f8dsfald om \u00e5ret.   Der er kun udviklet f\u00e5 nye antibiotika i l\u00f8bet af det sidste \u00e5rti, og de fleste er sm\u00e5 justeringer af eksisterende antibiotika.  Det er us\u00e6dvanligt arbejdskr\u00e6vende at opdage nye l\u00e6gemidler, men i et nyt skels\u00e6ttende studie har man udnyttet kunstig intelligens til automatisk at screene tusindvis af stoffer for at afd\u00e6kke muligheder for laboratorietest.  I unders\u00f8gelsen, som blev offentliggjort i Nature Chemical Biology, fors\u00f8gte forskere fra MIT og McMaster University at finde nye l\u00e6gemidler til at dr\u00e6be Acinetobacter baumannii,<\/p>","protected":false},"author":2,"featured_media":951,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[84],"tags":[105,101],"class_list":["post-950","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-industry","tag-machine-learning","tag-medtech"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>AI discovers new antibiotic for drug-resistant bacteria | DailyAI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" 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